Publications
of Patrick J. Bednarski
2011
Wasilewska, A., Saczewski, F., Gdaniec, M., Makowska, A., Bednarski, P.J. (2011) Synthesis of highly functionalized tetrahydropyridines with potential biological activity. Archive of Organic Chemistry (ARKIVOC), Part (x): 160-181.
Buczkowska, M. Bodtke, A., Lindequist, U., Gdaniec, M.,
Bednarski, P.J. (2011) Cytotoxic and antimicrobial
activities of Cu(II), Co(II), Pt(II) and Zn(II) complexes with N,O-chelating heterocyclic
carboxylates. Archiv der Pharmazie
Riechert-Krause, F., Eick, A., Grünert, R., Bednarski, P.J., Weisz, K. (2011) In vitro anticancer activity and evaluation of DNA duplex binding affinity of phenyl-substituted indoloquinolines. Bioorganic & Medicinal Chemistry Letters 21: 2380-2383.
Pomarnacka, E., Kornicka, A.,
Kuchnio, A., Heinrichs, M., Grünert, R., Gdaniec, M., Bednarski, P.J. (2011) Synthesis,
cytotoxicity testing and structure activity relationships of novel
6-chloro-7-(4-phenylimino-4H-3,1-benzoxazin-2-yl)-3-(substituted)-1,4,2-benzodithiazine
1,1-dioxides. Archiv der Pharmazie 344: 431-441.
Grünert,
R., Westendorf, A., Buczkowska, M., Hänsch, M., Kühne, S., Bednarski, P.J. (2011)
Cytotoxicity Testing-Cell Experiments. In : Metallointercalators
(J. Aldrich-Wright, Ed.) Springer Verlag, Wien ( ISBN: 978-3-211-09427-3).
Westendorf, A., Bodtke, A.,
Bednarski, P.J. (2011) Studies on the photoactivation of two cytotoxic
trans,trans,trans-diazidodiaminodihydroxo-Pt(IV) complexes.
Saczewski, J, Gdaniec, M.,
Bednarski, P.J., Makowska, A. (2011) Synthesis of aza-aromatic hydroxylamine-O-sulfonates
and their application to tandem nucleophilic addition-electrophilic 5-endo-trig
cyclization. Tetrahedron 67: 3612-3618.
Westendorf, A., Zerzankova, L.,
Salassa, L., Sadler, P.J., Brabec, V., Bednarski, P.J. (2011) Influence of pyridine versus
piperidine ligands on the chemical, DNA binding and cytotoxic properties of light
activated trans,trans,trans-[Pt(N3)2(OH)2(NH3)(L)]. Journal of Inorganic
Biochemistry 105: 652-662.
2010
Salassa, L., Ruiu, T., Garino, C.,
Pizarro, A. M., Bardelli, F., Gianolio, D., Westendorf, A., Bednarski, P. J., Lamberti,
C., Gobetto, R., Sadler, P. J. (2010) EXAFS, DFT, Light-Induced Nucleobase
Binding, and Cytotoxicity of the Photoactive Complex cis-[Ru(bpy)2(CO)Cl]+. Organometallics
29: 6703-6710.
Sunnam, S. K., Schepmann, D., Rack,
E., Froehlich, R., Korpis, K., Bednarski, P. J., Wuensch, B. (2010) Synthesis and
biological evaluation of conformationally restricted s1
receptor ligands with 7,9-diazabicyclo[4.2.2]decane scaffold. Organic &
Biomolecular Chemistry 8: 5525-5540.
Saczewski,
F., Kuchnio, A., Samsel, M., Lobocka, M., Kiedrowska, A., Lisewska, K., Saczewski, J.,
Gdaniec, M., Bednarski, P.J. (2010) Synthesis of novel aryl(heteroaryl)sulfonyl ureas of
possible biological interest. Molecules. 15: 1113-1126.
Reszka, P.,
Schulz, R., Methling, K., Lalk, M., Bednarski, P.J. (2010) Synthesis, enzymatic evaluation
an docking studies of fluorogenic caspase 8 tetrapeptide substrates. ChemMedChem
5: 103-117. (See journal
frontcover!)
2009
Holl,R., Jung, B., Schepmann, D.,
Humpf, H-U, Grünert, R, Bednarski P.J.,Englberger, Wünsch, W. (2009) Synthesis and
pharmacological evaluation of SNC80 analogues with a bridged piperazine ring. ChemMedChem
4: 2111-2122
Mothana R.A.A., Jansen, R.,
Grünert, R., Bednarski, P.J., Lindequist, U. (2009) Antimicrobial and cytotoxic abietane
diterpenoids from the roots of Meriandera benghalesis (Roxb.) Benth. Pharmazie
64: 613-615.
Kornicka, A., Hudson, A.L.,
Bednarski, P.J. (2009) Synthesis and biological activity of some 2-imidazolinylhydrazone
derivates. Acta Poloniae Pharmaceutica 66: 523-534.
Krause-Heuer, A.M., Grünert, R.,
Kühne, S., Buczkowska, M., Wheate, N.J., Le Pevelen, D.D., Boag, L.R., Fisher, D.M.,
Kasparkova, J., Malina, J., Bednarski, P.J., Brabec, V., Aldrich-Wirght, J.R. (2009)
Studies of the mechanism of action of platinum(II) complexes with potent cytotoxicty in
human cancer cells. Journal of Medicinal Chemistry 52: 5474-5484.
Bertrand, H., Bombard, S., Monchaud,
D., Talbot, E., Guedin, A., Mergny, J.-L., Grünert, R., Bednarski, P.J., Teulade-Fichou,
M.-P. (2009) Exclusive
platination of loop adenines in the human telomeric G-quadruplex. Organic and
Biomolecular Chemistry 7: 2864 - 2871.
Olszewski, U., Ach, F., Ulsperger,
E., Baumgartner, G., Zeillinger, R., Bednarski, P., Hamilton, G. (2009) In
vitro-evaluation of oxoplatin, an oral platinum(IV) anticancer agent. Metal-Based
Drugs. Article ID 348916
Hamberger, J., Liebeke, M., Kaiser,
M., Bracht, K., Olszewski, U., Zeillinger, R., Hamilton, G., Braun, D., Bednarski, P.J.
(2009) Characterisation of chemosensitivity and resistance of human cancer cell lines to
platinum (II) versus platinum(IV) anticancer agents. Anti-Cancer Drugs 20:
559-572
Mothana, R., Lindequist, U.,
Grünert, R., Bednarski, P.J. (2009)
Studies of the in vitro anticancer, antimicrobial and antioxidant potentials of selected
Yemeni medicinal plants from the island Soqotra. BMC
Complementary and Alternative Medicine 9: 7
Willemann, C., Grünert, R.,
Bednarski, P.J., Troschütz, R. (2009) Synthesis and cytotoxicity activity of
5,6-heteroaromatically annulated pyridine-2,4-diamines. Bioorganic & Medicinal
Chemistry 17: 4406-4419.
Holl, R., Schepmann, D., Fröhlich,
R, Grünert, R., Bednarski, P.J., Wünsch, B. (2009) Dancing of the second aromatic
residue around the 6,8-diazabicyclo[3.2.2]nonane framework: influence on receptor affinity
and cytotoxicity. Journal of Medicinal Chemistry
Kornicka, A., Bednarski, P.J. (2009)
Reaction of 2-chloro-4,5-dihydroimidazole with 1-aminobenzimidazoles: Synthesis of novel
fused heterocyclic ring systems. Polish Journal of Chemistry 83: 693-696.
Mothana, R., Grünert, R.,
Bednarski, P., Lindequist, U. (2009) Evaluation of the in vitro anticancer, antimicrobial
and antioxidant activities of some Yemeni plants used in the folk medicine. Pharmazie 64: 260-268.
Pomarnacka, E., Kornicka, A.,
Bednarski, P.J., Charkiewicz, A. (2009) Syntheses of N,S-Substituted
4-chloro-2-mercapto-5-merthylbenzensulfonamide derivatives with potential biological
activity. Polish Journal of Chemistry 83: 65-73.
Mendoza-Ferri, M., Hartinger, C.,
Mendoza-Parra, M., Groessl, M., Egger, A., Eichinger, R., Mangrum, J., Farrell, N.,
Maruszak, M., Bednarski, P., Klein, F., Jakupec, M., Nazarov, A., Severin, K., Keppler, B.
(2009) Transferring the concept of multinuclearity to ruthenium complexes for improvement
of anticancer activity. Journal of Medicinal Chemistry 52: 916-925.
Holl, R., Schepmann, D., Bednarski,
P.J., Grünert, R., Wünsch, B., (2009) Relationships between the structure of
6-substituted 6,8-diazabicyclo[3.2.2]nonan-2-ones and their sigma-receptor affinity and
cytotoxic activity.
Holl, R., Schepmann, D., Grünert,
R., Bednarski, P.J., Wünsch, B., (2009)
Methling K., Reszka, P., Lalk,
M., Vrana, O., Scheuch, E., Siegmund, W., Terhaag, B., Bednarski, P.J. (2009)
Investigations of the in vitro metabolism of the analgesic flupirtine. Drug Metabolism
and Disposition. 37: 479-493.
2008
Willemann, C., Waibel, R., Grünert,
R., Bednarski, P., Troschütz, R. (2008) Unexpected formation of pyridodiindole derivates
with cytotoxic activity via double Nenitzescu reaction. Journal of Heterocyclic
Chemistry 45:1517-1519..
Ruf, S., Neudert, G., Gürtler, S.,
Grünert, R., Bednarski, P.J., Otto, H.-H. (2008) ß-Lactam derivatives as potential
anti-cancer compounds. Monatshefte für Chemie 139: 847-857.
Saczewski, F., Stencel, A.,
Bienczak, A.M., Langowska, K.A., Michaelis, M., Werel, W., Halasa, R., Reszka, P.,
Bednarski, P.J. (2008) Structure activity relationships of novel heteroaryl-acrylonitriles
as cytotoxic and antibacterial agents. European Journal of Medicinal Chemistry 43:
1847-1857.
Pomarnacka, E., Maruszak, M.,
Langowska, K., Reszka, P., Bednarski, P.J. (2008) Synthesis and cytotoxicity testing of
novel 2-(3-substituted-6-chloro-1,1-dioxo -1,4,2-benzodithiazin-7-yl)-3-phenyl-4(3H)-quinazolinones.
Archiv der Pharmazie 341: 485-490.
Vogel, S., Kaufmann, D., Pojarova,
M., Müller, C., Pfaller, T., Kühne, S., Bednarski, P.J., von Angerer E. (2008) Aroyl
hydrazones of 2-pheylindole-3-carbaldehydes as novel antimitoic agents, Bioorganic
& Medicinal Chemistry. 16: 6436-6447.
Libnow, S., Methling, K., Hein, M.,
Michalik, D., Harms, M., Wende, K., Flemming, A., Köckerling, M., Reinke, H., Bedanrski,
P.J., Lalk, M., Langer, P. (2008) Synthesis of indirubin-N'-glycosides and their
anti-proliferative activity against human cancer cell lines. Bioorganic &
Medicinal Chemistry 16: 5570-5583.
Saczewski, F., Maruszak, M.,
Bednarski, P.J. (2008) Synthesis and cytotoxic activity of imidazo[1,2-a]-1,3,5-triazine
analogues of 6-mercaptopurine. Archiv der Pharmazie 341: 121-125.
Reszka, P., Methling K., Lalk, M.,
Xiao, Z., Weisz, K., Bednarski, PJ. (2008) Control of aspartate epimerization during the
coupling of caspase specific tetrapeptides with aromatic amines by using
N-[[(dimethylamino)-1H-1,2,3-triazolo[4,5-b]-pyridin-1-yl]methylene]-N-methylmethanaminium
hexafluorophosphate N-oxide (HATU) as a coupling reagent. Tetrahedron: Asymmetry 19:
49-59.
2007
Geiger,
C., Zelenka, C., Weigl, M., Fröhlich, R., Wibbeling, B., Lehmkuhl, K.,
Schepmann, D., Grünert, R., Bednarski, P.J., Wünsch, B. (2007) Synthesis of bicyclic s receptor ligands with cytotoxic activity
Pojarová, M., Kaufmann, D.,
Gastpar, R., Nishino, T., Reszka, P., Bednarski P.J., von Angerer, E (2007) [(2-Phenylindol-3-yl)methylene]propanedinitriles inhibit the growth of breast
cancer cells by cell cycle arrest in G2/M phase and apoptosis. Bioorganic
& Medicinal Chemistry 15: 7368-7379.
Bracht, K., Kiefer, T., Doelken, G.,
Bednarski, P.J. (2007) Characterization of three B-cel lymphoma cell lines from
chemotherapy resistant patients with respect to in vitro senstitivity to 21 antitumor
agents, ABC-transporter experession and cellular redox status. Journal of Cancer
Chemotherapy and Clinical Oncology, 133: 957-967.
Saczewski, F., Dziemidowicz-Borys,
E., Bednarski, P.J. and Gdaniec, M.(2007) Synthesis, crystal structure, cytotoxic and
superoxide dismutase activities of copper(II) complexes of N-(4,5-dihydroimidazol-2-yl)azoles. Archiv der Pharmazie 340: 333-338.
Brzozowski, Z., Saczewski, F.,
Slawinski, J., Bednarski, P.J., Grünert, R., Gdaniec, M. (2007) Synthesis, structural
characterization, and in vitro antitumor activity of novel N-(6-chloro-1,1-dioxo-1,4,2-benzodithiazin-3-yl)arylsulfonamides.
Bioorganic & Medicinal
Chemistry 15: 2560-2572.
Mothana, R.A.A., Grünert, R.,
Lindequist, U., Bednarski, .PJ. (2007) Study of the anticancer potential of Yemeni plants
used in folk medicine. Pharmazie 62: 305-307.
Fisher, D.M., Bednarski,
P.J., Grünert, R., Turner, P., Fenton, R.R., Aldrich-Wright, J.R. (2007)
Chiral platinum(II) metallointercalators with potent in vitro cytotoxic activity. ChemMedChem
2: 488-495.
Bracht, K., Liebeke, M.,
Bednarski, P.J., Mackay,
F.S., Sadler, P.J. (2007) Photoactivatable platinum complexes. Anti-Cancer
Agents in Medicinal Chemistry 7: 75-93. (Review)
2006
Bracht, K., Boubakari, Grünert R.,
Bednarski P.J. (2006) Correlations between the activities of 19 antitumor agents and the
intracellular GSH concentrations in a panel of 14 human cancer cell lines: Comparisons
with the NCI data. Anti-Cancer Drugs 17: 41-51.
Bednarski, P.J., Grünert, R.,
Zielzki, M., Wellner, A., Mackay, F.S., Sadler, P.J. (2006) Light-activated cestruction of
cancer cell nuclei by platinum diazide complexes. Chemistry & Biology 13:
61-67 (see cover) (see
Nature Highlight) (read Faculty
of 1000 Biology expert opinion).
Saczewski F., Bulakowska, A.,
Bednarski P. Grünert R. (2006) Synthesis, structure and anticancer activity
of novel 2,4-diamino-1,3,5-triazine derivatives. European Journal of Medicinal
Chemistry 41: 219-225.
Pomarnacka, E., Bednarski, P.J., Reszka, P.,
Dyiemidowicz-Borys, E., Bienczak, A., Werel, W., Halasa, R. (2006) Synthesis and
biological activity of new
2-amino-8-chloro-5,5-dioxo[1,2,4]triazolo[2,3-b][1,4,2]benzodithiazines. European
Journal of Medicinal Chemistry 41: 633-639.
Pomarnacka, E., Bednarski, P.J., Grünert, R.,
Brzozowski, Z., Lach, J. (2006) Synthesis and in vitro cytotoxic activity of novel
6-chloro-1,1-dioxo-1,4,2-benzodithiazin-3-ylhydrazine derivatives. Polish Journal of
Chemistry 80: 429-438.
Saczewski, J., Brzozowski, Z., Saczewski, F., Bednarski,
P.J., Liebeke, M., Gdaniec, M. (2006) Synthesis and in vitro anti-tumor activity of
N-{1-8(3-thioxo-5,6-dihydroimidazo82,1-c][1,2,4]thiadiazol-7-ylthio)thiocarbaonyl]-2-imidazol-idene}-arylsulfonamides.
Bioorganic & Medicinal Chemistry Letters 16:
3663-3667.
Saczewski, F., Dziemidowicz-Borys, E., Bednarski, P.J.,
Grünert, R., Gdaniec, M., Tabin, P. (2006) Synthesis, crystal structure and biological
activities of copper(II) complexes with chelating bidentate 2-substituted benzimidazole
ligands. Journal of Inorganic Biochemistry 100:
1389-1398.
Bose, G., Bracht, K., Bednarski, P.J., Lalk, M., Langer,
P. (2006) Synthesis, reactions and structure-activity relationships of
1-hydroxysprio[2.5]cyclooct-4-en-3-ones: Illudin analogs with in vitro cytotoxic activity.
Bioorganic & Medicinal Chemistry 14: 4694-4703.
2005
Pomarnacka, E., Bednarski, P.,
Grünert, R., Reszka, P. (2005) Synthesis and anticancer activity of novel
2-amino-4-(4-phenylpiperazino)-1,3,5-traizine derivatives. Acta Poloniae Pharmaceutica
61: 461-466.
2004
Slawinski J., Bednarski P., Reszka
P. (2004): Syntheses and in vitro antitumor activity of
3-amino-N-(4-chlorobenzenesulfonyl)guanidine derivatieves containing N'-arylidene moiety. Polish
Journal of Chemistry 78: 369-380.
Saczewski, F., Reszka, P., Gdaniec,
M., Grünert, R., Bednarski, P.J. (2004) Synthesis, x-ray crystal structures, stabilities
and in vitro cytotoxic activities of new heteroaryl-acrylonitriles. Journal of
Medicinal Chemistry 47: 3438-3449.
2003
Slawinski J., Bednarski P., Gruenert
R., Reszka P. (2003): Syntheses of a new series of N-amino-N¢
-(benzenesulphonyl)guanidine derivatives with potential antitumor activity. Polish
Journal of Chemistry 77: 53-64.
Achilles, K., Bednarski, P.J.
(2003): Quantification of elastase-like activity in 13 human cancer cell lines and in an
immortalized human epithelial cell line by RP-HPLC. Biololgical Chemistry 384:
817-824.
Neumann, Ch., Boubakari, Grünert,
R., Bednarski, P.J. (2003) Nicotinamide adenine dinucleotide phosphate-regenerating system
coupled to a glutathione microtiter method for determination of total glutathione
concentrations in adherent growing cancer cell lines. Analytical Biochemistry
320: 170-178.
Kushev, D., Grünert,
R., Spassovska, N., Golovinsky, E., Bednarski, P.J. (2003) Unusual reactivity
of cytotoxic cis-dihydrazide Pt(II) complexes in aqueous solution. Journal of
Inorganic Biochemistry 96: 469-477.
2001
Rinke, K., Grünert, R., Bednarski,
P.J. (2001): New synthetic route to [bis-1,2-(aminomethyl)benzene]dichloroplatinum(II)
complexes, screening for cytotoxic activity in cisplatin-sensitive and resistant human
cancer cell lines, and reaction with glutathione. Pharmazie 56: 763-769.
1999
Kratochwil, N. A., Parkinson, J. A., Bednarski, P. J. , Sadler,P. J. (1999): Platinierung von Nucleotiden, induziert durch sichtbares Licht. Angewandte Chemie 111: 1566-1569. (Press release!)
Kratochwil, N. A., Bednarski, P.
J. (1999): Relationships
between reduction properties and cancer cell growth inhibitory activities of cis-dichloro-
and -diiodo-Pt(IV)-ethylenediamines. Archiv der Pharmazie 332: 279-285.
Kratochwil, N. A., Bednarski,
P. J. (1999): Kinetics of thiol-release from human cancer
cells and their effects on the stability of Pt(IV)-complexes in culture medium. Journal
of Cancer Research and Clinical Oncology 125: 690-696.
Bednarski, P.J. (1999):
JM-216 Johnson Matthey plc. Current Opinion in Oncologic, Endocrine & Metabolic
Investigational Drugs 1: 448-458. (Review)
1998
Kratochwil, N. A., Guo, Z.,
1997
Mahboobi, S., Dove, S., Bednarski, P.J., Kuhr, S., Burgemeister, Th., Schollmeyer, D.
(1997): X-ray crystal structure of woodinine and conformational analysis by semiempircal
and 1H-NMR methods. Journal of Natural Products 60: 587 - 591.
1996
Köckerbauer, R., Bednarski, P.J. (1996): Unusual reactivity of cisplatin analogues that
bear o-phenylenediamine ligands: Insights for the design of more effective cytotoxic
agents. Journal of Inorganic Biochemistry 62: 281 - 298.
Kratochwil, N.A., Bednarski, P.J., Mrozek, H., Vogler, A., Nagle, J.K. (1996): Photolysis
of an iodoplatinum(IV) diamine complex to cytotoxic species by visible light. Anti-Cancer
Drug Design 11: 155 - 171.
Kratochwil, N.A., Zabel, M., Range, K.-J., Bednarski, P.J. (1996): Synthesis and X-ray
crystal structure of trans,cis-[Pt(OAc)2I2(en)]: A novel type of cisplatin analog
that can be photolyzed by visible light to DNA-binding and cytotoxic species in vitro. Journal
of Medicinal Chemistry 39: 2499 - 2507.
1995
Bednarski, P.J. (1995): Reactions of
a cisplatin analogue bearing an estrogenic 1,2-diarylethylenediamine ligand with
sulfur-containing amino acids and glutathione. Journal of Inorganic Biochemistry
60: 1 - 19.
Köckerbauer, R., Bednarski, P.J. (1995): A novel approach to preparing water soluble
prodrug-forms of cisplatin analogues bearing chelating diamines. Journal of
Pharmaceutical Sciences 84: 819 - 823.
Otto, A.M., Kratochwil, N.A., Eggers, H., Bednarski, P.J. (1995): Chemical stability,
biological activity and cellular uptake of a cisplatin analogue having a
1,2-diarylethylenediamine ligand in cultures of human breast cancer cells. Journal of
Cancer Research and Clinical Oncology 121: 31 - 38.
1994
Bednarski, P.J., Trümbach, B. (1994): Use of reversed-phase HPLC for the determination of
the hydrolysis rate constants of dichloro(1,2-diarylethylenediamine)platinum(II)
complexes. Transition Metal Chemistry 19: 513 - 517.
1993
Bednarski,P.J., Hartmann, R. (1993)
Synthesis and evaluation of sulfur-containing glutethimide derivatives for aromatase and
desmolase inhibitory activity. Archiv der Pharmazie, 326: 391-394.
1992
Otto, A.M., Bednarski, P.J., Eggers,
H., Trümbach, B., Schönenberger, H. (1992) [meso-1,2-Bis(2,6-dichloro-4-hydroxyphenyl)ethylenediamine]dichloroplatinum(II),
an estrogenic Pt(II)- complex for the therapy of breast cancer: relationship between
stability and effect. Pharmaceutical and Pharmacological Letters, 1: 103-106.
Müller,R., Bednarski, P.J.,
Schönenberger, H. (1992) (1,2-Diaryl-1,2-ethylenediamine)platin-um(II) complexes
with sulfato and 3-sulfopropionato leaving groups: investigations with differenttypes of
coordination in the solid state, in solution and reactions with nucleophiles. Inorganic
Chimica Acta, 195: 77-87.
Bednarski,P.J. (1992)
Relationships between the aqueous chemistry and the in vitro cytotoxic activities of
mixed-amine cisplatin analogues. Biochemical Pharmacology, 43: 2609-2620.
Bednarski,P.J., Trümbach, B.,
Kratochwil, N.A., Schönenberger, H. (1992) Diamine ligand release from the
cisplatin analogue [meso-1,2-Bis(2,6-dichloro-4-hydroxyphenyl)ethylenediamine]dichloroplatinum(II)
in cell culture medium. Journal of Medicinal Chemistry, 34: 4479-4485.
1991
Bednarski,P.J., Ehrensperger, E.,
Schönenberger, H., Burgemeister, T. (1991) Aqueous chemistry of mixed-amine cis- and
transplatin analogues. Intramolecular preference for a kineticsix-membered ring over a
thermodynamic five-membered ring ortho-platination product. Inorganic Chemistry,
30: 3015-3025.
1990
Bednarski,P.J., Gust, R., Spruß,
T., Knebel, N., Otto, A., Fardel, M., Koop, R., Holler, E., von Angerer, E.,
Schönenberger, H. (1990) Platinum compounds with estrogen receptor affinity. Cancer
Treatment Reviews, 17: 221-231.
1989
Bednarski,P.J., Nelson, S.D. (1989)
Interactions of thiol-containing androgens with human placental aromatase. Journal of
Medicinal Chemistry, 32: 203-213.
1985
Silvestri, M.G., Bednarski, P.J.,
Kho, E. (1985) Stereoselective insertion of the isopropenyl functionality. Journal
of Organic Chemistry, 50: 2798-2799.
1984
Nelson,W.L., Bartels, M.J.,
Bednarski, P.J., Zhang, S., Messick, K., Horng, J.S., Ruffolo, R.R. (1984) The
3,4-catechol derivative of propranolol, a minor dihydroxylated metabolite. Journal
of Medicinal Chemistry, 27: 857-861.
